GPCRProfiler Services
For quotes, please contact GPCRProfiler@millipore.com(Human unless noted) | ||||
| A | non-peptide | Acetylcholine (muscarinic) | M1 | |
| A | non-peptide | Acetylcholine (muscarinic) | M2 | |
| A | non-peptide | Acetylcholine (muscarinic) | M3 | |
| A | non-peptide | Acetylcholine (muscarinic) | M4 | |
| A | non-peptide | Acetylcholine (muscarinic) | M5 | |
| A | non-peptide | Adenosine | A1 | |
| A | non-peptide | Adenosine | A2B | |
| A | non-peptide | Adenosine | A3 | |
| A | non-peptide | Adrenergic | alpha1A | |
| A | non-peptide | Adrenergic | alpha1B | |
| A | non-peptide | Adrenergic | alpha1D | New |
| A | non-peptide | Adrenergic | alpha2A | |
| A | non-peptide | Adrenergic | alpha2B | |
| A | non-peptide | Adrenergic | beta 1 | |
| A | non-peptide | Adrenergic | beta 2 | |
| A | non-peptide | Adrenergic | beta 3 | |
| A | non-peptide | alpha-Ketoglutarate | OXGR1 , GPR99 , GPR80 | |
| A | peptide | Anaphylotoxin | C3aR | |
| A | peptide | Anaphylotoxin | C5aR | |
| A | peptide | Angiotensin | AT1 | |
| A | peptide | Apelin | APJ | New |
| A | peptide | Bombesin | BB1 | |
| A | peptide | Bombesin | BB2 | |
| A | peptide | Bombesin | BB3 | |
| A | peptide | Bradykinin | B2 | |
| B | peptide | Calcitonin | CGRP1 | |
| C | non-peptide | Calcium sensor | CaS | |
| A | non-peptide | Cannabinoid | CB1 | |
| A | non-peptide | Cannabinoid | CB2 | |
| A | peptide | Chemoattractant | ChemR23 / CMKLR1 | |
| A | peptide | Chemokine | CCR1 | |
| A | peptide | Chemokine | CCR10 | |
| A | peptide | Chemokine | CCR2B | |
| A | peptide | Chemokine | CCR3 | |
| A | peptide | Chemokine | CCR4 | |
| A | peptide | Chemokine | CCR5, rhesus macaque | |
| A | peptide | Chemokine | CCR6 | |
| A | peptide | Chemokine | CCR7 | |
| A | peptide | Chemokine | CCR8 | |
| A | peptide | Chemokine | CCR9 | |
| A | peptide | Chemokine | CX3CR1 | |
| A | peptide | Chemokine | CXCR1 / IL-8a | |
| A | peptide | Chemokine | CXCR2 / IL-8b | |
| A | peptide | Chemokine | CXCR3 | |
| A | peptide | Chemokine | CXCR4 | |
| A | peptide | Chemokine | CXCR5 | Coming Soon |
| A | peptide | Chemokine | CXCR6 | New |
| A | peptide | Chemokine | XCR1 / GPR5 | |
| A | peptide | Cholecystokinin | CCK1 / CCKa | |
| A | peptide | Cholecystokinin | CCK2 / CCKb | |
| B | peptide | CRF Receptor | CRF1 | |
| B | peptide | CRF Receptor | CRF2 | |
| A | non-peptide | Dopamine | D1 | |
| A | non-peptide | Dopamine | D2L | |
| A | non-peptide | Dopamine | D4 | Coming Soon |
| A | non-peptide | Dopamine | D5 | |
| A | peptide | Endothelin | ETA | |
| A | peptide | Endothelin | ETB | |
| A | non-peptide | Free Fatty Acid | FFA1 / GPR40 | |
| A | non-peptide | Free Fatty Acid | FFA2 / GPR41 | |
| A | non-peptide | Free Fatty Acid | FFA3 / GPR43 | |
| C | non-peptide | GABAB | GABAB1b | |
| A | peptide | Galanin | GAL1 | |
| A | peptide | Galanin | GAL2 | |
| A | peptide | Ghrelin | Ghrelin / GHSR-1a / growth hormone secretagogue receptor | New |
| B | peptide | Glucagon | GIP | |
| B | peptide | Glucagon | GLP-1 | |
| B | peptide | Glucagon | glucagon / GCG | |
| B | peptide | Glucagon | secretin receptor / SEC | |
| C | non-peptide | Glutamate (metabotropic) | mGlu2 | New |
| A | peptide | Glycoprotein hormone | TSH / TSHR | New |
| A | peptide | GnRH | GnRH / LHRH | |
| A | non-peptide | Histamine | H1 | |
| A | non-peptide | Histamine | H2 | |
| A | non-peptide | Histamine | H3 | |
| A | peptide | KiSS1-derived peptide | KiSS1 / GPR54 | |
| A | non-peptide | Leukotriene | BLT1 | |
| A | non-peptide | Leukotriene | CysLT1 | |
| A | non-peptide | Leukotriene | CysLT2 | |
| A | non-peptide | Lysophospholipid | LPA1 / EDG2 | |
| A | non-peptide | Lysophospholipid | LPA3 / EDG7 | |
| A | non-peptide | Lysophospholipid | GPR92 / LPA5 | New |
| A | non-peptide | Lysophospholipid | S1P1 / EDG1 | |
| A | non-peptide | Lysophospholipid | S1P2 / EDG5 | |
| A | non-peptide | Lysophospholipid | S1P3 / EDG3 | |
| A | non-peptide | Lysophospholipid | S1P4 / EDG6 | |
| A | non-peptide | Lysophospholipid | S1P5 / EDG8 | |
| A | peptide | Mas-related gene | MRGX1 / MRGPRX1 | New |
| A | peptide | Mas-related gene | MRGX2 / MRGPRX2 | |
| A | peptide | Mas-related gene | MRGPRD / MrgD | New |
| A | peptide | Melanin-concentrating hormone | MCHR1 / GPR24 | |
| A | peptide | Melanin-concentrating hormone | MCHR2 | |
| A | peptide | Melanocortin | MC2 | |
| A | peptide | Melanocortin | MC4 | |
| A | peptide | Melanocortin | MC5 | |
| A | peptide | Motilin | motilin receptor / MTLR / GPR38 | |
| A | peptide | Neuromedin U | NMU1 | |
| A | peptide | Neuromedin U | NMU2 | New |
| A | peptide | Neuropeptide B/W | NPBW1 / GPR7 | |
| A | peptide | Neuropeptide Y | Y2 | |
| A | peptide | Neuropeptide Y | Y4 | |
| A | peptide | Neurotensin | NTR1 / NTS1 | |
| A | peptide | N-formylpeptide | FPR1 | |
| A | peptide | N-formylpeptide | FPRL1 / AXL / HM63 | |
| A | non-peptide | Nicotinic Acid | GPR109A | |
| A | peptide | Opioid | Delta / OP1 / DOP / DOR | |
| A | peptide | Opioid | Kappa / OP2 / KOP / KOR | |
| A | peptide | Opioid | Mu / OP3 / MOP / MOR | |
| A | peptide | Opioid | NOP / ORL1 / OP4 | |
| A | peptide | Orexin | OX1 | |
| A | peptide | Orexin | OX2 | |
| A | peptide | Oxytocin | OT | |
| A | non-peptide | P2 / Purinergic (metabotropic) | P2Y1 | |
| A | non-peptide | P2 / Purinergic (metabotropic) | P2Y2 | New |
| A | non-peptide | P2 / Purinergic (metabotropic) | P2Y4 | New |
| A | non-peptide | P2 / Purinergic (metabotropic) | P2Y11 | New |
| A | peptide | Peptide P518 | GPR103 / QRFP | |
| A | non-peptide | Platelet Activating Factor | PAF | |
| A | peptide | Prokineticin | PK1 / PKR1 | |
| A | peptide | Prokineticin | PK2 / PKR2 | |
| A | peptide | Prolactin-releasing peptide | PRP / PrRP / GPR10 | |
| A | non-peptide | Prostanoid | DP | |
| A | non-peptide | Prostanoid | EP1 | |
| A | non-peptide | Prostanoid | EP2 | |
| A | non-peptide | Prostanoid | EP3 | |
| A | non-peptide | Prostanoid | EP4 | |
| A | non-peptide | Prostanoid | FP | |
| A | non-peptide | Prostanoid | IP1 / PGI2 | |
| A | non-peptide | Prostanoid | TP / TXA2 / PGH2 | |
| A | peptide | Protease-activated | Thrombin-activated PARs | |
| A | peptide | Protease-activated | Trypsin-activated PARs | |
| B | peptide | PTH receptor | PTH1 | |
| B | peptide | PTH receptor | PTH2 | |
| A | non-peptide | Serotonin | 5-HT1A | |
| A | non-peptide | Serotonin | 5-HT2A | |
| A | non-peptide | Serotonin | 5-HT2B | |
| A | non-peptide | Serotonin | 5-HT2C | |
| A | non-peptide | Serotonin | 5-HT6 | Coming Soon |
| A | peptide | Somatostatin | sst2 | |
| A | peptide | Somatostatin | sst3 | |
| A | peptide | Somatostatin | sst4 | |
| A | peptide | Somatostatin | sst5 | |
| A | non-peptide | SPC/LPC /proton-sensor | GPR68/OGR1 | |
| A | peptide | Tackykinin /neurokinin | NK1 | |
| A | peptide | Tackykinin /neurokinin | NK2 | |
| A | peptide | Tackykinin /neurokinin | NK3 | |
| A | peptide | TRH | TRH | |
| A | peptide | Urotensin II | UT / UT1 / GPR14 | |
| A | peptide | Vasopressin | V1A | |
| A | peptide | Vasopressin | V1B | |
| A | peptide | Vasopressin | V2 | |
| B | peptide | VIP/PACAP | PAC1 long isoform / PACAP | |
| B | peptide | VIP/PACAP | VPAC1 / VIP1 | |
| B | peptide | VIP/PACAP | VPAC2 / VIP2 |
